Cart
sales@molnova.com
Isoetharine mesylate salt
CAS No. 7279-75-6
Isoetharine mesylate salt( Isoetarine mesilate )
Catalog No. M19891 CAS No. 7279-75-6
Isoetharine Mesylate Salt is a β-adrenergic receptor agonist. it also is pregnane X receptor (PXR) activator capable of upregulating CYP450 expression.
Purity : >98% (HPLC)
COA
Datasheet
HNMR
HPLC
MSDS
Handing Instructions
| Size | Price / USD | Stock | Quantity |
| 25MG | 42 | In Stock |
|
| 50MG | 53 | In Stock |
|
| 100MG | 76 | In Stock |
|
| 200MG | Get Quote | In Stock |
|
| 500MG | Get Quote | In Stock |
|
| 1G | Get Quote | In Stock |
|
Biological Information
-
Product NameIsoetharine mesylate salt
-
NoteResearch use only, not for human use.
-
Brief DescriptionIsoetharine Mesylate Salt is a β-adrenergic receptor agonist. it also is pregnane X receptor (PXR) activator capable of upregulating CYP450 expression.
-
DescriptionIsoetharine Mesylate Salt is a β-adrenergic receptor agonist. it also is pregnane X receptor (PXR) activator capable of upregulating CYP450 expression.(In Vitro):Isoetharine mesylate (50 μM, 18 hours) can induce the production and release of [35S]sulfated metabolites of catecholic drugs in HepG2 human hepatoma cells.(In Vivo):Isoetharine mesylate inhibits melanin deposition with the AC50 value of 5.10 mM and complete inhibition of pigment production at 7.50 mM in the zebrafish larvae model.
-
In VitroIsoetharine mesylate (50 μM, 18 hours) can induce the production and release of [35S]sulfated metabolites of catecholic drugs in HepG2 human hepatoma cells.
-
In VivoIsoetharine mesylate inhibits melanin deposition with the AC50 value of 5.10 mM and complete inhibition of pigment production at 7.50 mM in the zebrafish larvae model.
-
SynonymsIsoetarine mesilate
-
PathwayAngiogenesis
-
TargetAdrenergic Receptor
-
Recptorβ-adrenergic receptor| PXR
-
Research AreaOthers
-
Indication——
Chemical Information
-
CAS Number7279-75-6
-
Formula Weight335.42
-
Molecular FormulaC14H25NO6S
-
Purity>98% (HPLC)
-
SolubilityDMSO:199.7 mM;Water:199.7 mM
-
SMILESCS(O)(=O)=O.CCC(NC(C)C)C(O)c1ccc(O)c(O)c1
-
Chemical Name——
Shipping & Storage Information
-
Storage(-20℃)
-
ShippingWith Ice Pack
-
Stability≥ 2 years
Reference
1.Ratajewski M et al. Screening of a chemical library reveals novel PXR-activating pharmacologic compounds. Toxicol Lett. 2015 Jan 5;232(1):193-202.
molnova catalog
related products
-
Dicentrine
Dicentrine is a natural product isolated from the plant Lindera megaphylla with antihypertensive effect. Dicentrine is an α1-adrenoceptor antagonist which has effective against human hyperplastic prostates.
-
ARC 239 dihydrochlor...
A potent, selective α2B adrenoceptor antagonist with pKd of 8.8, 200-fold selectivity over α2A, and α2D receptors.
-
BRL 44408 maleate
A potent, selective α2A-adrenoceptor antagonist with Ki of 1.7 nM, 80-fold selectivity over α2B-adrenergic receptors.
