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Isoetharine mesylate salt
CAS No. 7279-75-6
Isoetharine mesylate salt( Isoetarine mesilate )
Catalog No. M19891 CAS No. 7279-75-6
Isoetharine Mesylate Salt is a β-adrenergic receptor agonist. it also is pregnane X receptor (PXR) activator capable of upregulating CYP450 expression.
Purity : >98% (HPLC)
COA
Datasheet
HNMR
HPLC
MSDS
Handing Instructions
| Size | Price / USD | Stock | Quantity |
| 25MG | 42 | In Stock |
|
| 50MG | 53 | In Stock |
|
| 100MG | 76 | In Stock |
|
| 200MG | Get Quote | In Stock |
|
| 500MG | Get Quote | In Stock |
|
| 1G | Get Quote | In Stock |
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Biological Information
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Product NameIsoetharine mesylate salt
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NoteResearch use only, not for human use.
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Brief DescriptionIsoetharine Mesylate Salt is a β-adrenergic receptor agonist. it also is pregnane X receptor (PXR) activator capable of upregulating CYP450 expression.
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DescriptionIsoetharine Mesylate Salt is a β-adrenergic receptor agonist. it also is pregnane X receptor (PXR) activator capable of upregulating CYP450 expression.(In Vitro):Isoetharine mesylate (50 μM, 18 hours) can induce the production and release of [35S]sulfated metabolites of catecholic drugs in HepG2 human hepatoma cells.(In Vivo):Isoetharine mesylate inhibits melanin deposition with the AC50 value of 5.10 mM and complete inhibition of pigment production at 7.50 mM in the zebrafish larvae model.
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In VitroIsoetharine mesylate (50 μM, 18 hours) can induce the production and release of [35S]sulfated metabolites of catecholic drugs in HepG2 human hepatoma cells.
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In VivoIsoetharine mesylate inhibits melanin deposition with the AC50 value of 5.10 mM and complete inhibition of pigment production at 7.50 mM in the zebrafish larvae model.
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SynonymsIsoetarine mesilate
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PathwayAngiogenesis
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TargetAdrenergic Receptor
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Recptorβ-adrenergic receptor| PXR
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Research AreaOthers
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Indication——
Chemical Information
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CAS Number7279-75-6
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Formula Weight335.42
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Molecular FormulaC14H25NO6S
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Purity>98% (HPLC)
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SolubilityDMSO:199.7 mM;Water:199.7 mM
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SMILESCS(O)(=O)=O.CCC(NC(C)C)C(O)c1ccc(O)c(O)c1
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Chemical Name——
Shipping & Storage Information
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Storage(-20℃)
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ShippingWith Ice Pack
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Stability≥ 2 years
Reference
1.Ratajewski M et al. Screening of a chemical library reveals novel PXR-activating pharmacologic compounds. Toxicol Lett. 2015 Jan 5;232(1):193-202.
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